Direct Decarboxylative Giese Addition of Unprotected Amino Acids: A Cascade Access to γ-Lactams

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ID: 313714
2026
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Abstract
Abstract Unprotected amino acids were developed as precursors of α-aminoalkyl radicals under visible-light photoredox catalysis. Single-electron oxidation of deprotonated amino acids followed by decarboxylation generated α-amino radicals, which participated in intermolecular Giese-type additions to electron-deficient alkenes. The reaction proceeds without protection of the amino group and provides direct access to secondary and tertiary amine frameworks. The free amino functionality also enables a cascade process in which the initially formed adduct undergoes intramolecular cyclization to afford γ-lactam products. Electrochemical analysis and control experiments support a mechanism involving base-assisted oxidation of the amino acid and subsequent radical generation. This study establishes an efficient strategy for the generation and utilization of α-aminoalkyl radicals from readily available amino acids and demonstrates their utility in C–C bond formation.
Reference Key
openalex_W7160963364 Use this key to autocite in the manuscript while using SciMatic Manuscript Manager or Thesis Manager
Authors Tomotoki Matsuo, Yuto Sumida, Hirohisa Ohmiya
Journal bulletin of the chemical society of japan
Year 2026
DOI
10.1093/bulcsj/uoag058
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