Biomimetic Enantioselective Total Synthesis of (-)-Robustanoids A and B and Analogues.

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ID: 238215
2019
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Abstract
We report a step-economical, enantioselective total synthesis of (-)-robustanoid B and (-)-robustanoid A and four novel natural product-like compounds. Our strategy relied on our biosynthetic hypothesis and on a novel complexity generation methodology, namely, the one-pot hydroxylative double cyclization reaction. The latter consists of a modified 3,3-dimethyldioxirane-triggered epoxidation-epoxide-ring-opening cyclization reaction cascade and Trost's regioselectivity umpolung methodology ("anti-Michael addition").
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liu2019biomimeticthe Use this key to autocite in the manuscript while using SciMatic Manuscript Manager or Thesis Manager
Authors Liu, Zhan-Jiang;Huang, Pei-Qiang;
Journal The Journal of organic chemistry
Year 2019
DOI
10.1021/acs.joc.9b00573
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